Voatinggine and tabertinggine, pentacyclic indole alkaloids derived from an iboga precursor via a common cleavamine-type intermediate.

نویسندگان

  • Choy-Eng Nge
  • Chew-Yan Gan
  • Yun-Yee Low
  • Noel F Thomas
  • Toh-Seok Kam
چکیده

Two new indole alkaloids, voatinggine (1) and tabertinggine (2), which are characterized by previously unencountered natural product skeletons, were isolated from a Malayan Tabernaemontana species. The structures and absolute configuration of these alkaloids were determined using NMR and MS analysis, and X-ray diffraction analysis. A possible biogenetic pathway to these novel alkaloids from an iboga precursor, and via a common cleavamine-type intermediate, is presented.

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عنوان ژورنال:
  • Organic letters

دوره 15 18  شماره 

صفحات  -

تاریخ انتشار 2013